Organic & biomolecular chemistry

(ISSN: 1477-0520, 1477-0539)

Table of Contents

2014 - 12 (11)

  • Lead identification and structure-activity relationships of heteroarylpyrazole arylsulfonamides as allosteric CC-chemokine receptor 4 (CCR4) antagonists. 
  • Towards the diastereoselective synthesis of derivative of 11'-epi-brevipolide H. 
  • Ligand mediated iron catalyzed dimerization of terminal aryl alkynes: scope and limitations. 
  • Synthesis of 3-acyltetramates by side chain manipulation and their antibacterial activity. 
  • Copper-catalyzed decarboxylative C3-acylation of free (N-H) indoles with α-oxocarboxylic acids. 
  • Dissecting non-covalent interactions in oxazaborolidinium catalyzed cycloadditions of maleimides. 
  • Porphyrin conjugated with serum albumins and monoclonal antibodies boosts efficiency in targeted destruction of human bladder cancer cells. 
  • Transmembrane anion transport and cytotoxicity of synthetic tambjamine analogs. 
  • Efficient synthesis of functionalized dihydroquinolines, quinolines and dihydrobenzo[b]azepine via an iron(III) chloride-catalyzed intramolecular alkyne-carbonyl metathesis of alkyne tethered 2-amino benzaldehyde/acetophenone derivatives. 
  • Chemical synthesis of staphyloferrin A and its application for Staphylococcus aureus detection. 
  • Principles of modern solid-phase oligosaccharide synthesis. 
  • Catalytic regioselective synthesis of pyrazole based pyrido[2,3-d]pyrimidine-diones and their biological evaluation. 
  • Water promoted C-C bond cleavage: facile synthesis of 3,3-bipyrrole derivatives from dienones and tosylmethyl isocyanide (TosMIC). 
  • Unexpected regio- and chemoselectivity of cationic gold-catalyzed cycloisomerizations of propargylureas: access to tetrasubstituted 3,4-dihydropyrimidin-2(1H)-ones. 
  • Targeting abasic site-containing DNA with annelated quinolizinium derivatives: the influence of size, shape and substituents. 
  • Rh-catalyzed oxidative C-C bond formation and C-N bond cleavage: direct access to C2-olefinated free (NH)-indoles and pyrroles. 
  • Sequential stereodivergent organocatalysis and programmed organocascades. 
  • Synthesis of the tumor associative α-aminooxy disaccharide of the TF antigen and its conjugation to a polysaccharide immune stimulant. 
 
 

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